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This pipeline identified 6 known and 43 novel CRBN–pomalidomide binders, including orthogonally validated hits
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« Plus la dose est élevée, moins elle est absorbée » À faibles ou moyennes doses, également appelées doses physiologiques – celles que l’on apporte par l’alimentation (y compris, dans ce contexte, la B12 provenant d’aliments enrichis ou de suppléments à très faibles doses) –, l’absorption dépend du facteur intrinsèque sécrété et des récepteurs intestinaux du complexe de Castle, qui régulent ce processus
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